Tecarfarin (ATI-5923) is an orally active and non-competitive vitamin K epoxide reductase (VKOR) antagonist. It impairs the activation of the vitamin K-dependent clotting factors II, VII, IX, and X, demonstrating antithrombotic activity.
- Orally active
- Non-competitive VKOR antagonist
- Impairs activation of vitamin K-dependent clotting factors II, VII, IX, and X
- Has antithrombotic activity
- Solid appearance
- White to off-white color
- Soluble in DMSO at 250 mg/mL